T7665

Tyrphostin 51

≥98%

• 동의어(들): 2-Amino-1,1,3-tricyano-4-(3′,4′,5′-trihydroxyphenyl)butadiene
• 실험식(Hill 표기법): C₁₃H₈N₄O₃
• CAS Number: 126433-07-6
• Molecular Weight: 268.23
• MDL number: MFCD00133903
• UNSPSC 코드: 12352200
• PubChem Substance ID: 24278756
• NACRES: NA.77

속성

• 생물학적 소스: synthetic (organic)
• Quality Level: 200
• 분석: ≥98%
• 양식: powder
• 효능: 0.8 μM IC₅₀
• solubility: DMSO: soluble 5 mg of Tyrphostin 51 in 0.1 ml of solvent, clear, orange to red
• 저장 온도: 2-8°C
• SMILES string: NC(\C(=C\c1cc(O)c(O)c(O)c1)C#N)=C(/C#N)C#N
• InChI: 1S/C13H8N4O3/c14-4-8(12(17)9(5-15)6-16)1-7-2-10(18)13(20)11(19)3-7/h1-3,18-20H,17H2/b8-1+
• InChI key: JKNOYWVMHPMBEL-UNXLUWIOSA-N
• 유전자 정보: human ... CDK2(1017), EGFR(1956)

설명

애플리케이션

Tyrphostin 51 has been used to study the inhibition of rat hepatic leptin 1.

생화학적/생리학적 작용

EGFR tyrosine kinase inhibitor.

Tyrphostin 51 is a small molecule inhibitor of epidermal growth factor (EGF) receptor kinase function. This molecule associates with the substrate subsite of the protein tyrosine kinase (PTK) domain,.

특징 및 장점

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제조 메모

5 mg of Tyrphostin 51 is soluble in 0.1 ml of DMSO and yields a clear, orange to red solution.

안전성 정보

• Storage Class Code: 11 - Combustible Solids
• WGK: WGK 3
• Flash Point (°F): Not applicable
• Flash Point (°C): Not applicable
• 개인 보호 장비: Eyeshields, Gloves, type N95 (US)