PZ0229

PF-03246799 hydrochloride

≥98% (HPLC)

• 동의어(들): 6,7,8,9-Tetrahydro-2-(phenylmethyl)-5H-pyrimido[4,5-d]azepine hydrochloride, PF-3246799 hydrochloride
• 실험식(Hill 표기법): C₁₅H₁₇N₃ · xHCl
• CAS Number: 1065114-52-4
• Molecular Weight: 239.32 (free base basis)
• UNSPSC 코드: 51111800
• PubChem Substance ID: 329823781
• NACRES: NA.77

속성

• Quality Level: 100
• 분석: ≥98% (HPLC)
• 양식: powder
• 색상: white to beige
• solubility: H₂O: 20 mg/mL, clear
• 저장 온도: room temp
• SMILES string: C1(CC2=NC(CCNCC3)=C3C=N2)=CC=CC=C1.Cl
• InChI: 1S/C15H17N3.ClH/c1-2-4-12(5-3-1)10-15-17-11-13-6-8-16-9-7-14(13)18-15;/h1-5,11,16H,6-10H2;1H
• InChI key: ICVPRIZGSIUCOE-UHFFFAOYSA-N

설명

생화학적/생리학적 작용

PF-3246799 is a potent serotonin 5-HT2C receptor agonist with an EC₅₀ of 4.5 nM and minimal activity at 5-HT2A and 5-HT2B receptors. PF-3246799 had good efficacy in a preclinical canine model of stress urinary incontinence.

PF-3246799 is a potent serotonin 5-HT2C receptor agonist.

특징 및 장점

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안전성 정보

• Storage Class Code: 11 - Combustible Solids
• WGK: WGK 3
• Flash Point (°F): Not applicable
• Flash Point (°C): Not applicable